Factional Potency:Dermorphin yog qhov tseem muaj zog dua li morphine. Kev tshawb fawb kwv yees nws yog30-50 lub sij hawm ntau zog tshaj morphineThaum muab cov tswj hwm intracerebrovularly (ncaj qha rau hauv lub hlwb ventricles) hauv cov qauv qws. Txawm tias peripherally, nws ua rau pom muaj potency.
● D - amino acid tus yuam sij:Lub d - ala residue tsis yog - sib ceg rau kev ua. Cov hluavtaws hluavtaws nrog l - Ala tau zoo tsis nyob hauv. Qhov no d - cov amino acid ua rau dermorths (enzymes uas tawg rau nws lub sijhawm ntev ntawm kev ua piv rau kev ua kom zoo sib xws.
● Cov siab siab - opioid receptor xaiv:Thaum nws tuaj yeem cuam tshuam nrog Delta thiab Kappa receptors nyob rau ntau dua qhov siab, dermorphin nthuav qhia qhov xav tau thiab muaj ib qho siab rau cov mu {}} opioid receptor. Qhov kev xaiv no ua rau nws lub zog ua piv txwv thiab kev zoo siab.
● Metabolic Stability:Lub d - Ala ala thiab c-}}}}}} ح{ល against tiv thaiv nws cov nqaij ntshav thiab cov ntaub so ntswg piv rau cov enkephats. Qhov no pab txhawb rau ib nrab - lub neej tshaj li ntau peptides.
● Ntshav free -} Barrier (BBB) Penetration:Txawm hais tias yog peptide, dermorphin qhia tau zoo heev rau kev nkag mus ntawm BBB, qhov tsis tshua muaj neeg rau peptides. Qhov no yog ib nrab ntaus nqi rau nws lipophilic (rog- soluble) cov yam ntxwv thiab muaj peev xwm ua kom muaj kev thauj khoom hauv nruab nrab cov hom phiaj zoo tom qab kev tswj hwm.
Hom - Cov teebmeem:Nws cov txiaj ntsig txiaj ntsig yog feem ntau pom hauv cov tsiaj yug menyuam. Nyob rau hauv nws cov qav fog hosts, nws txoj haujlwm yog kwv yees kom muaj kev tiv thaiv (deterring predators (tiv thaiv tus kheej lub luag haujlwm ntawm amphibians lub luag haujlwm hauv amphibians tsis tau txhais.
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