Tirzepatide yogtsisib tug peptide hormones, tab sis aSynthetic, Ib Leeg - saw 39-amino acid peptideengineered rau ua haujlwm raws li aLwl tag nrho - kav insulinottropic polypetropic polypepropic (Glucagon {(gpp-1) receptor agonistCov. Qhov no yog nws txoj kev txhais lus thiab txawv txav los ntawm ua ntej GLP-1-tsuas yog agonists xws li semaglutide.
● Kev siv tshuab:Tirzepatide tsis yog tsuas ua kom ob qho tib si receptors sib npaug; Kev tshawb fawb qhia tias nws muaj siab duaib qho muaj ib qho muaj ib qho affinityRau lub gip receptor tshaj qhov glp - 1 receptor. Lub synergistic nyhuv ntawm co-actemting cov pathways ua lub luag haujlwm rau nws qhov kev ua tau zoo hauv cov kab mob GLP-1 hauv kev sim tshuaj. Gip receptation yuav muaj lub zog ntawm cov txiaj ntsig ntawm GLP-1, tshwj xeeb rau kev noj qab haus huv thiab tej zaum muaj rog metabolism.






