Sildenafil Citrate

CAS: 171599-83-0
MF: C28H38N6O11S
wb: 666.7
Synonyms:, Sildenafil citrate;1-[[3-(6,7-Dihydro-1-methyl-7-oxo-3-propyl-1H-pyrazolo[4,3-d]pyrimidin-5-yl)-4-ethoxyphenyl]sulfonyl]-4-methylpiperazine, 2-hydroxy-1,2,3-propanetricarboxylate;1-[[3-(4,7-Dihydro-1-methyl-7-oxo-3-propyl-1H-pyrazolo[4,3-d]pyrimidin-5-yl)-4-ethoxyphenyl]sulfonyl]-4-methylpiperazine citrate salt;5-[2-Ethoxy-5-(4-methylpiperazin-1-yl)sulfonylphenyl]-1-methyl-3-propyl-4H-pyrazolo[5,4-e]pyrimidin-7-one citrate salt;Sildenafil Citrate (100 mg);Sildenafil citrate, >=99 feem pua ;Sildenafil citrate, Kev muab khoom;5-[2-Ethoxy-5-[(4-methyl-piperazin-1-yl)sulfonyl]phenyl ]-1,6-dihydro-1-methyl-3-propyl-7H-pyrazolo[4,3-d]pyrimidin-7-ib citrate
COA
| Cov khoom | Txuj | Cov txiaj ntsig |
| Kev ntsuam xyuas los ntawm HPLC: | 98 feem pua | 99.37% ua |
| Qhov tsos: | Dawb hmoov zoo | Ua raws |
| Cov ntxhiab thiab saj: | Me ntsis iab | Ua raws |
| Mesh loj: | 100% dhau 80 mesh | Ua raws |
| Solubility: | Soluble hauv dej | Ua raws |
| Loss ntawm ziab: | Tsawg dua lossis sib npaug rau 2.0 feem pua | 1.15 feem pua |
| Heavy hlau PPM: | <30ppm | Ua raws |
| Microbiology: Tag Nrho Plate Count: Pwm & Pwm: E.Coli: S. Aureus: Salmonella: |
<1000cfu/g <100cfu/g Tsis zoo Tsis zoo Tsis zoo |
800 cfu/g 90 cf/g Ua raws Ua raws Ua raws |
| Xaus: | Ua raws li USP 32 | |
Kev piav qhia
Sildenafil citrate yog ib hom tshuaj uas feem ntau siv los kho erectile kawg (ED) hauv cov txiv neej. Nws tseem raug muag raws li lub npe Viagra, thiab lwm yam. Sildenafil belongs rau ib chav kawm ntawm cov tshuaj hu ua phosphodiesterase type 5 (PDE5) inhibitors, uas ua haujlwm los ntawm kev ua kom cov ntshav ntws mus rau qhov chaw mos, pab txhawb kev erection thaum muaj kev sib deev stimulation.
Kev kho erectile kawg: Sildenafil citrate feem ntau yog muab rau kev kho mob ntawm erectile kawg, ib qho mob tshwm sim los ntawm kev tsis muaj peev xwm ua tiav lossis tswj kev erection txaus rau kev sib deev txaus siab. Nws muaj txiaj ntsig zoo hauv feem ntau ntawm cov xwm txheej, tsis hais qhov tshwm sim ntawm ED.
Mechanism of action: Sildenafil citrate ua haujlwm los ntawm inhibiting qhov kev txiav txim ntawm enzyme phosphodiesterase type 5 (PDE5). Qhov no inhibition nce qib ntawm cyclic guanosine monophosphate (cGMP), ib qho tshuaj uas ua kom cov leeg du hauv cov hlab ntsha ntawm tes. Qhov kev so no tso cai rau kom muaj ntshav ntau ntxiv mus rau qhov chaw mos, ua rau muaj erection thaum muaj kev sib deev stimulation.
Kev noj tshuaj thiab kev siv: Sildenafil citrate feem ntau yog noj hauv qhov ncauj, hauv daim ntawv ntsiav tshuaj, li 30 feeb mus rau 1 teev ua ntej kev sib deev. Cov tshuaj muaj txiaj ntsig tuaj yeem kav ntev txog li ob peb teev, muab lub sijhawm rau kev sib deev. Nws yog ib qho tseem ceeb uas yuav tsum tau ua raws li cov lus qhia thiab kev siv tshuaj uas tau muab los ntawm koj tus kws kho mob.
Teb thiab kev ua tau zoo: Sildenafil citrate tau pom tias muaj txiaj ntsig zoo rau feem coob ntawm cov txiv neej uas muaj erectile kawg. Txawm li cas los xij, cov lus teb ntawm tus kheej yuav txawv, thiab nws yuav tsis ua haujlwm rau txhua tus. Nws yog ib qho tseem ceeb rau kev sib txuas lus nrog koj tus kws kho mob txog qhov ua tau zoo ntawm cov tshuaj thiab txhua qhov kev hloov kho uas yuav xav tau.
Kev ceev faj thiab kev txiav txim siab: Ua ntej siv sildenafil citrate, nws yog ib qho tseem ceeb kom nthuav tawm koj cov keeb kwm kho mob thiab lwm yam tshuaj uas koj noj rau koj tus kws kho mob. Qee yam kev mob nkeeg, xws li teeb meem plawv, kab mob siab lossis raum, lossis keeb kwm ntawm priapism (ntev ntev thiab mob erection), yuav tsum tau ceev faj tshwj xeeb lossis kev hloov pauv ntau npaum li cas. Tsis tas li ntawd, sildenafil citrate yuav tsum tsis txhob siv nrog nitrates, vim qhov no tuaj yeem ua rau cov ntshav siab poob qis.
Kev mob tshwm sim: Cov kev mob tshwm sim feem ntau ntawm sildenafil citrate tuaj yeem muaj xws li mob taub hau, yaug, qhov ntswg congestion, plab zom mov, thiab kiv taub hau. Cov kev mob tshwm sim no feem ntau yog mob me thiab ntuav. Txawm li cas los xij, yog tias koj ntsib cov kev mob tshwm sim hnyav lossis ntev erections ntev tshaj li plaub teev (priapism), nrhiav kev kho mob tam sim ntawd.
Dosage thiab siv:
Sildenafil citrate, feem ntau paub los ntawm nws lub npe Viagra, yog cov tshuaj siv los kho erectile kawg (ED) hauv cov txiv neej. Nws ua haujlwm los ntawm kev ua kom cov ntshav ntws mus rau qhov chaw mos, pab kom ua tiav thiab tswj kev erection. Nov yog qee cov ntaub ntawv hais txog kev noj tshuaj thiab kev siv sildenafil citrate:
Kev siv:
Noj sildenafil citrate nrog ib khob dej. Tsis txhob noj nrog zaub mov hnyav, vim qhov no yuav ncua qhov pib ntawm nws cov teebmeem.
Sildenafil citrate ua haujlwm zoo tshaj plaws thaum muaj kev sib deev stimulation. Nws tsis ua rau tsis siv neeg erection.
Cov tshuaj feem ntau pib ua haujlwm li ntawm 30 mus rau 60 feeb tom qab noj, tab sis nws tuaj yeem sib txawv ntawm ib tus neeg mus rau lwm tus.
Cov teebmeem ntawm sildenafil citrate tuaj yeem kav ntev li plaub mus rau rau teev. Txawm li cas los xij, lub sijhawm tuaj yeem cuam tshuam los ntawm cov yam ntxwv xws li cov metabolism, kev noj qab haus huv tag nrho, thiab lwm yam tshuaj noj.
Tsis txhob noj sildenafil citrate yog tias koj tseem siv nitrates (xws li nitroglycerin) rau mob hauv siab lossis yog tias koj muaj qee yam mob. Nrog koj tus kws kho mob lossis tus kws muag tshuaj kom paub tseeb tias nws muaj kev nyab xeeb rau koj noj.
Nws yog ib qho tseem ceeb uas yuav tau tham nrog koj tus kws kho mob ua ntej pib sildenafil citrate los tham txog koj cov keeb kwm kev kho mob, txhua yam tshuaj uas koj tab tom noj tam sim no, thiab tej zaum muaj contraindications lossis kev phiv.
Txhua yam kev xav tau, thov hu rau kuv
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