YK11 yog dab tsi?
YK11 yog qhov tseeb tshaj plaws hauv lub hlis nyob rau hauv kev lag luam av grey kev ua lag luam tsim kho lub ntiaj teb. YK11 yog ib qho tshuaj stero molecule uas tsuas tau pom tias muaj cov teebmeem hauv kev ua haujlwm ntawm cellular. Qhov no txhais tau hais tias tseem tsis muaj kev tshaj tawm cov tsiaj lossis tib neeg tseem tsis tau tshwm sim. Txawm li ntawd los nws tau plaws tawm rau hauv kev muag khoom hauv is taws nem anabolic SARM lossis SARM.
Lub hnub nyoog tshiab SARMs zoo li LGD-4033 thiab Ostarine yog non-stero, lub ntsiab lus hais tias lawv tsis muaj plaub lub nplhaib qub qauv ntawm classical androgens zoo li Stero zoo li Nan thiab kab tias tre yuav suav tau tias yog SARMs txij thaum lawv hloov los ntawm 5-alpha txo rau tsawg zog androgens thiab hauv cov koob tshuaj tsim nyog qhia ntau dua anabolic dua li cov teebmeem androgenic. Stero tau hloov mus rau hauv cov lus tsis zoo yog li rau feem ntau, cov tuam txhab tab tom txhim kho SARMS tsis-stero. Hauv kev muaj tiag, nws ua rau me ntsis qhov sib txawv ntawm cov duab ntawm cov duab tab sis theej nws cov teebmeem yog li cas.
YK11 yog stero. Qhov tseeb, nws zoo li ntau. Ob daim ntawv uas muaj nyob ntawd qhia tias YK11 tuaj yeem qhib lub androgen receptor tab sis nws tsuas yog ua qee tus. Qhov no ua rau cov nyhuv paub li ib nrab agonism. Qhov no txhais tau hais tias YK11 tuaj yeem tshem tawm cov muaj zog androgens thaum muaj kev txo qis ntawm tag nrho cov kev cuam tshuam ntawm lub receptor. Qhov tseeb daim ntawv los ntawm Kanno et al ua kom pom cov nyhuv no los ntawm kev da dej hlwb hauv DHT ib leeg lossis hauv DHT + YK11. Cov hlwb uas tau txais ob qho DHT thiab YK11 muaj qhov kev xav androgenic tsawg dua nrog DHT ib leeg. Qhov no tseem ceeb vim tias, thaum muaj cov androgens muaj zog, YK11 yuav ua tau txo qhov androgen receptor stimulation. Kev ua rau prostate lossis plaub hau, qhov no tuaj yeem yog qhov ua tau zoo. Hauv cov leeg pob txha, qhov no yuav tsis yog qhov zoo.
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Cim npe nrov: sarms hmoov yk 11, Tuam Tshoj, tuam ntxhab, cov chaw muag khoom, lub Hoobkas, cov nqi teev, hauv Tshuag, cov qauv dawb












