tshuaj active cov khoom xyaw,tshuaj zoo tshuaj |
Cov ntsiab lus ceev
| Khoom npe | Ipamorelin |
| Synonyms | IpoMarelin; IpaMorelin Acetate; Aib-His-D-2-Nal-D-Phe-Lys-NH2;170851-70-4 |
| CAS | 170851-70-4 |
| MF | C38H49N9O5 |
| MW | 711.863 |
| MS | |
| EINECS | N/A |
| Yam khoom | Peptides |
| Qhov tshwm sim | Dawb Lyophilized Hmoov |
| Purity | 99 feem pua |
| Specification | 2 mg / vial |
| Cia | Lyophilized Ipamorelin ruaj khov ntawm chav tsev kub rau 90 hnub; txawm li cas los xij nws yuav tsum tau muab khaws cia rau hauv lub freezer hauv qab no -8C rau ib lub sij hawm ntev. Tom qab rov tsim dua, Ipamorelin yuav tsum tau muab tso rau hauv tub yees ntawm qhov kub tsis tshaj 36 F. |
| Kev siv | Ipamorelin yog ib qho kev xaiv loj hlob Hormone Secretagogue Thiab Agonist ntawm Ghrelin Receptor. |

Kev piav qhia
Ipamorelin yog qhov kev tshawb pom tshiab ntawm cov leeg nqaij zoo nkauj uas tau txais kev mloog ntau hauv ntiaj teb kev tsim lub cev. Nws yog ib qho hluavtaws peptide uas muaj zog loj hlob Hormone tso tawm cov khoom. Thiab cov GH tso tawm cov khoom no yog qhov txaus siab rau cov neeg ncaws pob thiab cov kws tsim lub cev vim lawv tuaj yeem ua qhov sib txawv ntawm cov leeg nqaij uas koj tuaj yeem loj hlob thiab koj hlawv rog sai npaum li cas.
Ipamorelin yog penta-peptide. (Aib-His-D-2-Nal-D- Phe-LysNH2) Thiab, lub zog uas nws qhia tau zoo heev ua rau cov laus hlob Hormone (GH) tsis siv. Tab sis dab tsi ncaws pob thiab bodybuilders xav paub yog dab tsi yog qhov xav tsis thoob peptide muaj peev xwm ua, nws siv li cas, thiab nws piv rau lwm yam GHRP peptides li cas?
Cov neeg ncaws pob tau noj Ipamorelin hauv ib koob tshuaj 200mcg300mcg, ob lossis peb zaug ib hnub, siv koob tshuaj insulin me me los txhaj. Lawv feem ntau pib nrog cov koob tshuaj qis dua txij li cov kev mob tshwm sim tuaj yeem muaj xws li mob taub hau lossis zoo li lub taub hau nrawm. Ipamorelin tuaj yeem noj tau txhua lub sijhawm tab sis noj nws li ntawm 30-45 feeb ua ntej kev tawm dag zog yuav zoo tagnrho vim tias cov mem tes hauv Growth Hormone (GH) nws tsim kom muaj kev loj hlob siab tshaj plaws.Studies txog cov teebmeem ntawm Ipamorelin ntawm cov pob txha loj hlob, lub cev qhov hnyav, thiab GH tso tawm tau pom qee qhov kev txiav txim siab nthuav dav.Nyob rau hauv ib qho kev sim, ntau cov koob tshuaj tau muab coj los siv rau hauv 15 hnub los ntsuam xyuas pab pawg cov tshuaj tiv thaiv.
Muaj qhov sib txawv thiab tsis muaj kev cuam tshuam rau lub cev qhov hnyav li cas los xij, pab pawg kho mob tsis pom qhov hloov pauv ntawm tag nrho IGFI qib. Tsis yog pab pawg kho mob tau tsim cov cim ntawm cov pob txha. Piv txwv li, tus naj npawb ntawm cov hlwb nyob rau hauv qhov dav ntawm tibia (lub shinbone) tsis hloov pauv loj. Qhov no yog qhov zoo vim hais tias nws qhia cov nqaij ntshiv uas tsis tshua muaj peev xwm rau deformity ntawm pob txha lossis pob txha mos.
Daim ntawv thov
Ipamorelin yog ib qho nthuav peptide noj 300mcg ob zaug ib hnub twg lossis koj tuaj yeem txo qhov koob tshuaj rau 3 zaug hauv ib hnub, cov kev mob tshwm sim yog mob taub hau, Kuv xav kom noj 30 feeb ua ntej kev tawm dag zog, nrog iav, Ipamorelin yog ib qho tshiab thiab muaj zog hluavtaws pentapeptide uas muaj qhov sib txawv thiab tshwj xeeb kev loj hlob hormone (GH)-tso cov khoom. Nrog rau lub hom phiaj ntawm kev soj ntsuam cov teebmeem ntawm cov pob txha ntev ntev, qhov hnyav ntawm lub cev, thiab GH tso tawm, Ipamorelin nyob rau hauv ntau koob tshuaj (0, 18, 90 thiab 450 ug / hnub) tau txhaj peb zaug ib hnub rau 15 hnub los ntsuas cov ntsiab lus, Tom qab intravital Tetracycline labeling rau hnub 0, 6, thiab 13, LGR tau txiav txim siab los ntawm kev ntsuas qhov kev ncua deb ntawm cov fluorescent bands nyob rau hauv proximal tibia metaphysis.
Ipamorelin koob tshuaj-raws li nce LGR ntawm 42 μm / hnub hauv pawg tsheb mus rau 44, 50, thiab 52 μm / hnub hauv pawg kho mob. Kuj tseem muaj qhov hais tawm thiab koob tshuaj raws li qhov tshwm sim ntawm lub cev qhov hnyav. Kev kho mob tsis cuam tshuam tag nrho IGF-I qib, lossis cov cim ntawm cov pob txha tsim thiab resorption. Tus naj npawb ntawm tartrate-resistant acid phosphatase-positive multinuclear hlwb hauv metaphysis ntawm tibia tsis hloov pauv nrog kev kho mob.
Ipamorelin tsis tsim pob hauv prolactin lossis cortisol zoo li GHRP-2 thiab -6. Ipa yog rab phom phom, tsis yog rab phom phom zoo li lwm tus GHRP. Tsis tas li ntawd nws yog qhov zoo rau cov neeg uas muaj calorie txwv tsis pub noj vim nws tsis txhawb kev qab los noj mov
Ipamorelin thiab Peptides yog txoj hauv kev ntawm lub neej yav tom ntej, cia siab tias nyob rau hauv 5 xyoo tom ntej los yog tsawg dua qhov kev hloov pauv loj hauv txoj kev uas peb cob qhia thiab coj lub ntiaj teb tsim lub cev los ntawm cua daj cua dub.
Muaj nuj nqi & Kev siv
Ipamorelin, zoo li lwm yam peptides, los ua cov hmoov qhuav qhuav uas muag heev. Koj tuaj yeem khaws cia rau hauv lub tub yees lossis hauv chav sov ua ntej rov tsim dua. Thaum rov tsim dua nrog dej bacteriostatic, cov vials yuav tsum tau muab cia rau hauv qhov chaw qhuav qhuav zoo li koj lub tub yees. Insulin syringes yog txoj hauv kev zoo tshaj plaws los tswj nws, feem ntau ntawm kev txhaj tshuaj subcutaneous.
Tau kawg, siv iPamorelin nrog GHRH zoo li CJC w/out DAC yuav ua rau tus neeg siv qhov loj tshaj ntawm GH thiab IGF-1 raws li GHRP's thiab GHRH ua haujlwm ua ke sib koom ua ke.
Qhov nruab nrab koob tshuaj rau Ipamorelin yog 200-300mcg ob mus rau peb zaug ib hnub twg. Kaum ob lub lis piam mus ncig yog qhov qub thiab PCT yuav tsawg heev - mini-pct zoo. Yog tias muaj teeb meem prolactin tshwm sim, muaj cov khoom uas pab txo qis prolactin thiab cov tsos mob zoo li estrogen. Cov no suav nrog aromatase inhibitors (Aromasin, Arimidex), thiab cov tshuaj tiv thaiv prolactin xws li Dostinex (Cabergoline).
Any xav tau, thov hu rau kuv
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