Cov lus piav qhia ntxaws ntxaws
| Qhov tsos: | Dawb rau lub teeb daj Crystalline hmoov | Lwm Lub Npe: | Fareston |
|---|---|---|---|
| Shipping Method: | EMS, HKEMS, FEDEX, DHL, UPS, Aramex, ETC | Stroage Temp: | 0-6 degree |
| MF: | C26H28ClNO | MW: | 598.09 |
| Lub teeb siab: | tshuaj tiv thaiv estrogen,anti estrogen khoom | ||
Abstract
Toremifene
Toremifene citrate yog lub qhov ncauj xaiv estrogen receptor modulator (SERM) uas pab tawm tsam cov kev ua ntawm estrogen hauv lub cev. Daim ntawv tso cai nyob rau hauv Tebchaws Meskas raws li hom npe Fareston, toremifene citrate yog FDA pom zoo siv rau kev mob qog noj ntshav siab (metastatic). Nws kuj tseem raug soj ntsuam rau kev tiv thaiv kab mob qog noj ntshav hauv qab lub npe Acapodene.
Dab tsi yog qhov zoo tshaj plaws steroid rau cov leeg nce?
Nws twb tau hais tias Toremifene yog SERM, thiab ua haujlwm los thaiv cov tshuaj Estrogen ntawm ntau qhov chaw receptors hauv qee cov ntaub so ntswg hauv lub cev (cov ntaub so ntswg ntawm lub mis tshwj xeeb). Raws li ib tug layman piav, Toremifene ua txuj ua ib tug 'fake' Estrogen uas occupies Estrogen receptors nyob rau hauv lub mis cov ntaub so ntswg. Nrog cov receptors nyob hauv Toremifene, tiag Estrogen tsis tuaj yeem ua lawv txoj haujlwm nyob ntawd.
Toremifene tsis txo tag nrho cov ntshav plasma qib ntawm Estrogen. Ntxiv rau qhov ua antagonistic rau Estrogen receptors nyob rau hauv lub mis cov ntaub so ntswg, nws kuj yog antagonistic rau Estrogen ntawm lub hypothalamus caj pas (qhov no tseem ceeb 'tricks' lub hypothalamus rau hauv kev xav muaj tsawg los yog tsis muaj circulating Estrogen theem nyob rau hauv lub cev, ua rau nws nce nws cov khoom. ntawm Testosterone kom nws tuaj yeem siv aromatization los kho cov qib no.

Toremifene kuj yog agonistic rau Estrogen receptors hauv lwm cov ntaub so ntswg hauv lub cev (hauv daim siab tshwj xeeb). Qhov no txhais tau hais tias thaum Toremifene yuav ua raws li cov tshuaj tiv thaiv estrogen hauv cov ntaub so ntswg ntawm lub mis thiab hypothalamus, nws yuav ua raws li Estrogen hauv daim siab. Qhov no tuaj yeem muaj txiaj ntsig zoo tshwj xeeb tshaj yog thaum lub voj voog anabolic steroid, xws li kev txhim kho thiab hloov cov qib roj cholesterol mus rau ntau qhov kev pom zoo.
Kev tswj hwm
Hauv kev sib ntaus tawm tsam mob qog noj ntshav mis, tus qauv Toremifene Citrate koob tshuaj yuav nquag yog 60mg ib hnub. Tag nrho lub sij hawm ntawm kev siv yog unpredictable thiab yuav ua raws li tus neeg mob xav tau. Nws tsis yog qhov nyuaj rau kev kho mob kom kav ib xyoos lossis ob xyoos thiab tom qab ntawd AI yuav tsum tau ntxiv yog tias xav tau. Thaum mob qog noj ntshav nyob rau hauv kev zam txim, cov tebchaw xws li Toremifene Citrate feem ntau yog siv los txhawb lub xeev txhim kho.
Rau cov neeg siv anabolic steroid combating gynecomastia, tus qauv Toremifene Citrate koob tshuaj yuav poob rau hauv 30-60mg ib hnub twg thiab yuav ua haujlwm zoo rau cov txiv neej feem ntau. Yog tias qhov no tsis muaj kev tiv thaiv txaus, thaum koj tuaj yeem sim nce koob tshuaj koj thawj koom ruam zoo tshaj plaws yuav txav mus rau AI siv. Koj yuav pom Toremifene Citrate ua haujlwm zoo heev hauv kev sib ntaus sib tua gynecomastia vim yog siv cov testosterone, Dianabol thiab Anadrol. Koj tseem yuav pom Toremifene Citrate ua haujlwm zoo nrog Equipoise thiab Deca Durabolin. Txawm li cas los xij, raws li Deca Durabolin kuj yog ib qho progestin, cov txiv neej uas nkag siab zoo rau cov tshuaj hormones no yuav xav tau AI. Tib yam tuaj yeem hais txog Trenbolone hormone.
Trenbolone tsis aromatize, tab sis nws yog ib tug progestin. Ntxiv mus, kev siv cov aromatizing steroid nrog ib tug compound zoo li Trenbolone tuaj yeem ua rau muaj kev pheej hmoo ntawm gynecomastia hauv qee tus txiv neej. Txawm hais tias ntau tus yuav tsis xav tau kev tiv thaiv gynecomastia vim yog progestins thiab yuav tau txais los ntawm SERM's los tawm tsam aromatase, qee tus txiv neej rhiab yuav xav tau AI. Txawm li cas los xij, yog tias Toremifene Citrate ua haujlwm rau koj, nws yuav npog tag nrho qhov dav ntawm lub voj voog txij thaum pib mus txog thaum xaus.
COA
| TEST ITEMSSPECIFICATIONRESULTSDEScriptionWhite los yog Yuav luag Dawb Dawb Crystalline PowderWhite PowderIdentificationPositivePositiveAssay97.00~103.00 feem pua 99.38 feem pua Pos Thaum ziab0.5 feem pua max{2{13}. feem pua Melting Point95~99¡ãC96.0~98.0¡ãCSpecific Rotation plus 48¡ã~ plus 51¡ã plus 49.0¡ãOrganic Volatile Impurities ua tau raws li qhov yuav tsum tau muaj.ConformsResidual Solvents ua tau raws li qhov yuav tsum tau muaj.Cov conformsConforms nrog USP32 tus qauv |
Cov txiaj ntsig
1. Nws muaj pov thawj hauv kev kho mob. Hauv ntau qhov kev ntsuas tseem ceeb ntawm cov tshuaj muaj txiaj ntsig hauv kev kho mob metastatic ER ntxiv rau kev mob qog noj ntshav mis hauv cov poj niam tom qab yug menyuam, Fareston tau ua haujlwm zoo li tamoxifen1-4
2. Tej zaum yuav muab cov txiaj ntsig txuas ntxiv ntawm kev kho mob endocrine. Fareston tuaj yeem muab cov txiaj ntsig txuas ntxiv rau koj ntawm kev kho mob endocrine yog tias koj tsis tuaj yeem zam lossis tsis tuaj yeem noj lwm yam kev kho mob endocrine1-6
3. Fareston tej zaum yuav yog ib txoj hauv kev zoo rau cov neeg mob uas tau tso tseg kev kho mob endocrine vim yog mob pob qij txha1-4,6
4. Muaj thiab siv tau. Fareston yog dav muaj nyob rau hauv kev lag luam thiab Medicare Part D cov qauv tsim thiab raug them los ntawm feem ntau kev lag luam thiab Medicare cov phiaj xwm pov hwm.

Kev noj tshuaj
Rau lub hom phiaj tsim lub cev, koob tshuaj 40-60mgs ib hnub zoo li yog qhov pib zoo. Yog tias tus neeg siv tab tom sim tawm tsam gynecomastia uas twb muaj lawm (bitch tits), lawv tuaj yeem xaiv ob npaug ntawm cov koob tshuaj thiab ntxiv ib qho aromatase inhibitor xws li Aromasin los ntawm kev siv nws. Rau PCT, ntau tus yuav pib nrog 100-120mgs txhua hnub thiab tom qab ntawd qis dua rau 40-60mgs txhua hnub rau 4-6 lub lis piam.
Yam khoom
| Anti-Estrogen | ||
| Tamoxifen Citrate (Nolvadex) | CAS: 54965-24-1 | |
| Clomiphene Citrate (Clomid) | CAS: 50-41-9 | |
| Toremifene Citrate (Fareston) | CAS: 89778-27-8 | |
| Femara | CAS: 112809-51-5 | |
| Aromasin | CAS: 107868-30-4 | |
| Proviron | CAS: 1424-00-6 | |
| Arimidex | CAS: 120511-73-1 | |
| Cabergoline (zeeg) | CAS: 81409-90-7 | |
| Finasteride | CAS: 98319-26-7 | |
| Dutasteride | CAS: 164656-23-9 | |
Txhua yam kev xav tau, thov hu rau kuv
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